CAS:212141-51-0|Vatalanib (PTK787) 2HCl
【产品介绍】:
产品名称 Vatalanib (PTK787) 2HCl 英文名称 Vatalanib (PTK787) 2HCl 规格或纯度 ≥99% 别名 瓦他拉尼二盐酸盐 英文别名 1-(4-Chloroanilino)-4-(4-pyridylmethyl)phthalazine dihydrochloride;CGP 79787 dihydrochloride;CGP 79787D dihydrochloride;N-(4-Chloroanilino)-4-(pyridin-4-ylmethyl)phthalazin-1-amine dihydrochloride;PTK787 dihydrochloride;ZK222584 dihydrochloride;Vatalanib 运输条件 超低温冰袋运输 生化机理 Vatalanib (PTK787) is a novel VEGFR and c-Kit tyrosine kinases and angiogenesis inhibitor with IC50 of 0.037, 0.077, 0.27 and 0.73 μM for KDR, Flt-1, Flk and c-Kit, respectively.Cell-permeable, potent, selective inhibitor of the VEGFR tyrosine kinases\xa0VEGFR-1 (Flt-1) and VEGFR-2 (FLK-1/KDR)\xa0(IC 50 values are 77 nM and\xa037 nM respectively).CAS编号 212141-51-0 溶解性 DMSO 85 mg/mL Water 10 mg/mL Ethanol 6 mg/mL 储存温度 -20°C储存 分子量 419.74 分子式 C20H15ClN4.2HCl 替代CAS 212141-54-3 PubChem CID 22386467